Free Fatty Acid Receptor (FFAR) (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-60167	GPR120 agonist 4x GPR120 (FFAR4) agonist	GPR120 agonist 4x is a potent, selective, orally bioavailable GPR120 agonist with EC50 of 42 nM in calcium flux assays.
PC-70042	DC-260126 GPR40 agonist	DC-260126 is a potent GPR40 agonist with IC50 of 6.28 uM for inhibition of Ca2+ stimulated by linoleic acid.
PC-42610	TAK-875 GPR40 agonist	TAK-875 (Fasiglifam) is a potent, selective, orally bioavailable GPR40 (FFA1) agonist with EC50 of 14 nM.
PC-42283	TUG-891 GPR120 (FFAR4) agonist	TUG-891 is a potent, selective human GPR120 (FFA4) agonist with pEC50 of 7.22.
PC-45843	GW-1100 GPR40 inhibitor	GW-1100 (SB-376752) is a potent, selective GPR40 antagonist that dose dependently inhibits GPR40-mediated Ca2+ elevations stimulated by GW9508 and linoleic acid with pIC50 of 5.99.
PC-45779	GSK137647A GPR120 (FFAR4) agonist	GSK-137647 (GSK-137647A) is a potent, selective GPR120 (FFA4) agonist with pEC50 of 6.3, >100-fold selectivity over the FFA1, FFA2, and FFA3 receptors.
PC-42400	GPR120 agonist 1 GPR120 (FFAR4) agonist	GPR120 agonist 1 is a potent, fully selective, orally available GPR120 (FFA4) agonist with pEC50 of 7.62.
PC-43813	AMG 837 GPR40 agonist	AMG 837 is a potent partial GPR40 (FFA1) agonist (EC50=13 nM for hGPR40).
PC-20869	GPR40 agonist AP4 GPR40 agonist	GPR40 agonist AP4 is a potent, selective, full allosteric agonist (AgoPAM) of GPR40 with EC50 of 0.08 nM, Emax=283%.

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