Formyl peptide receptor (FPR) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofFormyl peptide receptor (FPR) Formyl peptide receptor (FPR)

Cat. No.	Product Name	Information
PC-20394	BVT173187 FPR1 inhibitor	BVT173187 is a potent, selective, non-peptide inhibitor of formyl peptide receptor 1 (FPR1), inhibits fMLF and WKYMVM induced oxidase activity.
PC-20393	Quin-C1 FPR2 agonist	Quin C1 is a potent and selective FPR2 agonist with EC50 of 15 nM, induces Ca2+ mobilization in FPR2 but not FPR1-transfected mast cells.
PC-20392	HCH6-1 FPR1 inhibitor	HCH6-1 is a selective, competitive formyl peptide receptor 1 (FPR1) antagonist, superoxide anion generation in fMLF (FPR1 agonist)-activated neutrophils with IC50 of 0.32 uM in cell-impermeable cytochrome c reduction assay.
PC-20391	WRW4 FPR2 inhibitor	WRW4 (Trp-Arg-Trp-Trp-Trp-Trp) is a selective antagonist of formyl peptide receptor 2 (FPR2, FPRL1) signaling, inhibits WKYMVm binding to FPR2 with IC50 of 0.23 uM.
PC-49033	BMS-986235 FPR2 agonist	BMS-986235 (LAR-1219) is a potent, selective, and orally bioavailable agonist of formyl peptide receptor 2 (FPR2) with EC50 of 0.4 nM (hFPR2), >7,000-fold selectivity over FPR1.
PC-72355	FPR2 inhibitor (S)-11l FPR2 agonist	FPR2 inhibitor (S)-11l is a potent, selective, brain penetrant FPR2 agonist with IC50 of 0.13 uM (hFPR2).
PC-72086	FPR agonist Compound 43 FPR agonist	FPR agonist Compound 43 is a potent agonist of human formyl-peptide-like 1 receptor (hFPRL1) with EC50 of 44 nM (hFPRL1-mediated Ca2+ mobilization).
PC-72085	FPR agonist Compound 17b FPR agonist	FPR agonist Compound 17b is a small-molecule FPR1/FPR2 agonist withEC50 of 3.2 uM (hFPR1 Ca2+ mobilization), lack of functional responses at FPR3.
PC-72084	WKYMVm hexapeptide pan-FPR agonist	WKYMVm hexapeptide is a potent, selective, pan-agonist for the formyl peptide receptors FPR1, FPR2 (EC50 = 75 pM) and FPR3 (EC50 = 3 nM).
PC-72083	FPR1 agonist fMLF FPR1 agonist	FPR1 agonist fMLF (NSC 350593) is a potent, selective formylpeptide receptor-1 (FPR1) agonist with EC50 of 80 nM in calcium flux, Ki of 38 nM.
PC-72082	ICT12035 FPR1 antagonist	ICT12035 (AZ2158) is a potent, selective formylpeptide receptor-1 (FPR1) antagonist with IC50 of 30 nM in calcium mobilisation assays (100 nM fMLF).
PC-62594	ACT-389949 FPR2 agonist	ACT-389949 (ACT389949) is a novel potent and selective formyl peptide receptor type 2 (FPR2)/Lipoxin A4 receptor (ALX) agonist with EC50 of 3 nM for FPR2/ALX internalization into monocytes.

PREV12 NEXT