Dipeptidyl Peptidase (DPP) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofDipeptidyl Peptidase (DPP) Dipeptidyl Peptidase (DPP)

Cat. No.	Product Name	Information
PC-43412	Talabostat mesylate DPP4 inhibitor	Talabostat (PT-100, Val-boroPro) is a potent, nonselective, orally available inhibitor of post-proline cleaving serine proteases with Ki of 0.18 nM for DPP4, also potently inhibits DPP8/9 (IC50=1.5/0.76 nM), FAP, DPP2 and some other DASH family enzymes.
PC-43097	DBPR108 DPP4 inhibitor	Prusogliptin (DBPR108) is a potent, selective, orally bioavailable and long-acting inhibitor of DPP4 with IC50 of 15 nM, >3,000-fold selectivity over DPP8, DPP9, FAP and DPP-II.
PC-63161	AZD-5248 DPP-1 inhibitor	AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).
PC-61445	Evogliptin DPP-4 inhibitor	Evogliptin (DA1229) is a potent, long acting, reversible and competitive DPP-4 inhibitor with IC50 of 0.9 nM.
PC-60974	Gemigliptin DPP-4 inhibitor	Gemigliptin (LC15-0444) is a potent, selective, competitive and orally active DPP4 inhibitor (IC50=10.4 nM, hDPP4) with potential for the treatment of type 2 diabetes.
PC-60517	Gosogliptin dihydrochloride DPP-4 inhibitor	Gosogliptin dihydrochloride (PF-00734200) is a potent, selective, competitive, orally active dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 13 nM.
PC-60516	Gosogliptin DPP-4 inhibitor	Gosogliptin (PF-734200, PF-00734200) is a potent, selective, competitive, orally active dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 13 nM.
PC-60515	Garvagliptin DPP-4 inhibitor	Garvagliptin (NVP LAF 237A, LAF237A) is a potent, selective dipeptidyl peptidase-4 (DPP-4) inhibitor for treatment for type 2 diabetes.
PC-60064	Imigliptin dihydrochloride DPP-4 inhibitor	Imigliptin dihydrochloride (KBP-3853) is a potent, selective, orally available DPP-4 inhibitor with IC50 of 9 nM.
PC-44866	Omarigliptin DPP4 inhibitor	Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM.
PC-42508	Linagliptin DPP4 inhibitor	Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM.
PC-42510	Saxagliptin hydrate DPP4 inhibitor	Saxagliptin (BMS-477118) hydrate is a highly potent, long-acting, orally active DPP4 inhibitor with Ki of 0.6 nM.

PREV 123 NEXT