| Cat. No. |
Product Name |
Information |
| PC-22436 |
INDY
DYRK1A inhibitor
|
INDY is a potent, selective and ATP-competitive inhibitor of Dyrk1A withIC50 and Ki values of 0.24 and 0.18 μM, respectively. |
| PC-21660 |
Y020-3945
DYRK1A inhibitor
|
Y020-3945 is a selective dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitor with IC50 of 0.53 uM. |
| PC-21496 |
EHT 1610
DYRK1A inhibitor
|
EHT 1610 is a potent inhibitor of DYRKs family kinases with IC50s of 0.36 nM (DYRK1A), 0.59 nM (DYRK1B), respectively. |
| PC-21495 |
FC162
DYRK1A inhibitor
|
FC162 is a potent inhibitor of DYRK1A with IC50 of 11, 18, and 68 nM, against DYRK1A, CLK1, and GSK3, respectively. |
| PC-21494 |
EHT 5372
DYRK1A inhibitor
|
EHT 5372 is a highly potent and selective inhibitor of DYRKs family kinases with IC50s of 0.22, 0.28, 10.8, 93.2 nM for DYRK1A, DYRK1B, DYRK2, DYRK3, respectively. |
| PC-73294 |
MU1787
HIPK inhibitor
|
MU1787 is a potent, highly selective HIPK inhibitor with IC50 of 285/123/283 nM for HIPK1/2/3, repectively. |
| PC-73292 |
JWD-065
HIPK2 inhibitor
|
JWD-065 is a potent small molecule HIPK2 kinase inhibitor, blocks HIPK2 phosphorylation on S359/T360 and JNK activation in HEK293 cells and attenuates ER stress-induced cell death with EC50 of 641 nM. |
| PC-73291 |
CVM-6-139-1
HIPK2 inhibitor
|
CVM-6-139-1 (HIPK2 inhibitor A64) is a potent small molecule HIPK2 kinase inhibitor, blocks HIPK2 phosphorylation on S359/T360 and JNK activation in HEK293 cells and attenuates ER stress-induced cell death with EC50 of 401 nM. |
