| Cat. No. |
Product Name |
Information |
| PC-45775 |
MK-571 sodium salt
LTD4 inhibitor
|
MK-571 sodium is a potent and specific LTD4 receptor antagonist with Ki of 0.22 nM. |
| PC-23852 |
CAY10583
BLT2 agonist
|
CAY10583 is a potent and selective leukotriene B4 receptor type 2 (BLT2) agonist, inhibits LTB4 binding to BLT2 with IC50 of 20 nM, but not BLT1. |
| PC-23851 |
T-10430
BLT2 agonist
|
T-10430 is a potent and selective agonist of leukotriene B4 receptor 2 (BLT2) with EC50 of 0.51 nM in cAMP assays. |
| PC-23321 |
Pranlukast
CysLT antagonist
|
Pranlukast (SB 205312, ONO-1078) is a highly potent, selective and competitive leukotriene antagonist, inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Ki values of 0.63 nM, 0.99 nM, and 5640 nM, respectively. |
| PC-23320 |
Montelukast sodium
CysLT1 antagonist
|
Montelukast (MK0476) sodium is a potent, selective and orally active antagonist of cysteinyl leukotriene receptor 1 (CysLT1) with Ki of 0.18 nM, 4 nM and 0.52 nM in guinea pig lung, sheep lung and U937 cell plasma membrane preparations respectively. |
| PC-23319 |
Montelukast
CysLT1 antagonist
|
Montelukast (MK0476) is a potent, selective and orally active antagonist of cysteinyl leukotriene receptor 1 (CysLT1) with Ki of 0.18 nM, 4 nM and 0.52 nM in guinea pig lung, sheep lung and U937 cell plasma membrane preparations respectively. |
| PC-21194 |
U75302
LTB4 receptor 1 inhibitor
|
U75302 is a specific leukotriene B4 receptor 1 (LTB4 receptor 1, BLTR1, BLT1) inhibitor, effectively block LTB4 responses. |
