Cat. No. |
Product Name |
Information |
PC-61765 |
MRT199665
SIK inhibitor
|
MRT199665 is a potent salt-inducible kinases (SIKs) inhibitor with IC50 of 110, 12, 43 nM for SIK1,2,3 respectively. |
PC-42327 |
YKL-05-099
SIK inhibitor
|
YKL-05-099 (YKL 05-099) is a novel potent, selective pan-SIK inhibitor with IC50 of 10, 40 and 30 nM for SIK1, 2 and 3, respectively. |
PC-25119 |
SIK2-3 inhibitor 7s
SIK2/3 inhibitor
|
SIK2/3 inhibitor 7s is a potent, selective dual SIK2/3 inhibitor with IC50 of 1.1 nM for both, >30-fold selective over SIK1. |
PC-25118 |
GLPG4970
SIK2/3 inhibitor
|
GLPG4970 is a highly potent, selective dual SIK2/SIK3 inhibitor with IC50 of 0.3/0.7 nM respectively. |
PC-24280 |
SIK inhibitor 7s
SIK2/3 inhibitor
|
SIK inhibitor 7s is a potent, selective inhibitor of SIK2/SIK3 with IC50 of 1.1 nM for both, inhibits SIK1 with IC50 of 34.5 nM. |
PC-20809 |
SIK inhibitor M22
pan-SIK inhibitor
|
SIK inhibitor M22 is a potent, selective pan-SIK (salt-inducible kinase) with IC50 of 72, 89 and 18 nM for SIK1, SIK2 and SIK3 in NanoBERT assays, respectively. |