ROCK compound (inhibitors, antagonists, modulators)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-42540	Fasudil hydrochloride ROCK inhibitor	Fasudil hydrochloride (AT-877, HA-1077) is a potent and selective inhibitor of Rho kinase (ROCK) with Ki of 0.33 uM (ROCK1).
PC-42776	GSK429286A ROCK inhibitor	GSK429286A is a poten and selective inhibitor ROCK1 (IC50=14 nM) and ROCK2 (IC50=63 nM).
PC-27868	NRL-1049 dihydrochloride ROCK2 inhibitor	NRL-1049 dihydrochloride ((R)-BA-1049) is a potent, orally-available ROCK2-selective inhibitor with IC50 of 0.24 uM, 16-fold selectivity over ROCK-1.
PC-27410	Bazipsudil ROCK inhibitor	Bazipsudil is a potent, selective Rho-associated protein kinase (ROCK) inhibitor.
PC-25179	475A ROCK2 inhibitor	475A is a potent, highly selective ROCK2 inhibitor with IC50 of 1.3 nM, 162-fold selective over ROCK1 (IC50=211 nM).
PC-22511	GNS-3595 ROCK2 inhibitor	GNS-3595 is a potent and selective ROCK2 inhibitor with IC50 of 5.7 nM, 80-fold selectivity over ROCK1 at 1mM ATP.
PC-21755	C3TD879 Citron kinase inhibitor	C3TD879 is a potent, selective first-in-class Citron kinase (CITK) chemical inhibitor with biochemical IC50 of 12 nM.
PC-21300	ITRI-E-(S)4046 ROCK/MYLK4 inhibitor	ITRI-E-(S)4046 (E(S)4046) is a potent, highly specific, dual synergistic inhibitor of myosin light chain kinase 4 (MYLK4) and Rho-related protein kinase (ROCK) with IC50 of 3.2 nM and 25.6 nM for ROCK1 and MYLK4, respectively.

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