| Cat. No. |
Product Name |
Information |
| PC-43903 |
Olodaterol
β2 adrenoceptor agonist
|
Olodaterol (BI 1744) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
| PC-45155 |
Medetomidine
α2-adrenoceptor agonist
|
Medetomidine is a potent, highly selective α2-adrenoceptor agonist with Ki of 1.08 nM. |
| PC-45295 |
Carteolol hydrochloride
Beta-blocker
|
Carteolol hydrochloride is a non-selective beta-adrenoceptor antagonist (Beta-blocker) used as an anti-arrhythmia agent, an anti-angina agent, an antihypertensive agent, and an antiglaucoma agent. |
| PC-45270 |
Salmeterol
β2AR agonist
|
Salmeterol (GR33343X) is a long-acting beta2-adrenergic receptor agonist (Ki=1.5 nM) used clinically to treat asthma and maintenance of COPD. |
| PC-45299 |
Bambuterol hydrochloride
|
Bambuterol hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma. |
| PC-45298 |
Bambuterol
beta-adrenoceptor agonist
|
Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline. |
| PC-42338 |
Silodosin
α1A-adrenoceptor antagonist
|
Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM. |
| PC-27223 |
Alfuzosin hydrochloride
α1-adrenoceptor antagonist
|
Alfuzosin (SL 77499) hydrochloride is an orally active, selective and competitive α1-adrenoceptor antagonist, shows potential for prostatic hyperplasia (BPH). |
| PC-27222 |
Alfuzosin
α1-adrenoceptor antagonist
|
Alfuzosin (SL 77499) is an orally active, selective and competitive α1-adrenoceptor antagonist, shows potential for prostatic hyperplasia (BPH). |
| PC-27221 |
Doxazosin
α1-adrenoceptor antagonist
|
Doxazosin is a long-lasting, selective antagnist of α1-adrenoceptor antagonist receptors, shows potent apoptotic effect against prostate tumor epithelial cells, also has direct inhibitory effect on cholesterol synthesis independent of the LDL receptor. |
| PC-26994 |
SOM3355
β1-adrenergic receptor antagonist
|
Bevantolol hydrochloride (SOM3355) is a CNS-permeant, selective β1-adrenergic receptor antagonist with pKi value of 7.83 in rat cerebral cortex, also shows additional VMAT2 and VMAT1 inhibition activity. |
| PC-26836 |
Terazosin
PGK1 activator, α1-adrenergic receptor antagonist
|
Terazosin is a small molecule α1-adrenergic receptor antagonist and activator of phosphoglycerate kinase 1 (PGK1) at 2.5 nM -0.5 uM, binds to PGK1 with ITC Kd of 2.78 uM. |
