| Cat. No. |
Product Name |
Information |
| PC-26658 |
RX821002
α2A/D-adrenoreceptor antagonist
|
RX821002 (2-Methoxyidazoxan) is a highly selective antagonist of alpha2A/D-adrenoreceptor (alpha2A/D-AR) antagonist with pKd of 8.2 and 9.7 for rabbit alpha 2A-adrenoceptor and guinea-pig alpha 2D-adrenoceptor respectively. |
| PC-26581 |
A-61603
α1A AR agonist
|
A-61603 is a potent, selective alpha 1-adrenergic receptor (α1A AR) agonist, >35-fold more potent at α1A than at α1B or α1D sites, induces dose response increases in spontaneous Ca2+ transients in rat ventricular myocytes in vitro with EC50 of 6.9 nM. |
| PC-25621 |
Trifluoperazine
eEF2K inhibitor, α1-adrenergic receptor antagonist
|
Trifluoperazine is an antiadrenergic, antidopaminergic and anticholinergic agent, potent α1-adrenergic receptor antagonist, also inhibits calcium/calmodulin to eEF2K. |
| PC-25616 |
Vatinoxan hydrochloride
α2A adrenoceptor antagonist
|
Vatinoxan hydrochloride (MK-467, L-659066) is a potent and selective alpha-2 adrenoceptor (α2A adrenoceptor, α2AR) antagonist with IC50 of 3 nM against the binding of [3H]rauwolscine to rat cerebrocortical membranes, selective over alpha-1 adrenoceptors. |
| PC-25423 |
Formoterol fumarate
β2-adrenoceptor agonist
|
Formoterol fumarate is a potent, selective and long-acting β2-adrenoceptor agonist. |
| PC-25233 |
Imiloxan hydrochloride
α2B adrenoceptor antagonist
|
Imiloxan hydrochloride (RS 21361) is a potent and selective alpha 2B-adrenoceptor antagonist. |
| PC-25232 |
ADRIANA
α2B adrenoceptor antagonist
|
ADRIANA (c545) is a potent, orally active α2B adrenoceptor subtype-specific antagonist with binding Ki of 987 nM, >50-fold selective over α2A adrenoceptor. |
| PC-25231 |
ARC239
α2B adrenoceptor antagonist
|
ARC239 (ARC 239) is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-24801 |
Salbutamol
β2AR agonist
|
Salbutamol (Albuterol) is a, selective, orally active, short-acting beta-2 adrenergic receptor (β2AR) agonist, 29-fold more selective for beta2 receptors than beta1 receptors. |
| PC-24800 |
BRL-37344
β3AR agonist
|
BRL-37344 (BRL37344) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM. |
| PC-24569 |
Dabuzalgron
α1A-AR agonist
|
Dabuzalgron (Ro 115-1240) is an orally active and selective α-1A adrenergic receptor agonist with pKi of 7.39 for the displacement of [3H]-prazosin binding to CHO-K1 membranes. |
| PC-24491 |
Bisoprolol
β1AR antagonist
|
Bisoprolol is a second-generation, highly selective beta-1 adrenergic receptor (β1AR) antagonist with little activity on β2AR. |
