| Cat. No. |
Product Name |
Information |
| PC-25182 |
PAD-PF1
PAD inhibitor
|
PAD-PF1 is a small molecule potein arginine deiminase (PAD) inhibitor with binding KD of 2.82 uM and IC50 of 15.9 uM (PAD4). |
| PC-25181 |
PAD3 inhibitor 14b
PAD3 inhibitor
|
PAD3 inhibitor 14b is a potent and selective inhibitor of protein arginine deiminase PAD3 with kinact/KI value of 15600, ≥10-fold selectivity for PAD3 over PADs 1, 2, and 4. |
| PC-25180 |
AFM-30a hydrochloride
PAD2 inhibitor
|
AFM-30a hydrochloride is a potent, selective protein arginine deiminase 2 (PAD2) inhibitor with IC50 of EC50 of 9.5 uM in target engagement assays in HEK293/PAD2 cells. |
| PC-24593 |
PAD4 inhibitor GSK147
CAS 1549811-03-1
|
PAD4 inhibitor GSK147 is a potent, selective PAD4 inhibitor. |
| PC-23134 |
YW4-03
PAD4 inhibitor
|
YW4-03 is a small molecule peptidylarginine deiminase (PAD) inhibitor with IC50 of 5 uM against PAD4, exhibits cell-killing efficacy in osteosarcoma U2OS cells with IC50 of 2.5-5 uM. |
| PC-22866 |
Cl-amidine TFA
PAD inhibitor
|
Cl-amidine TFA is a potent, irreversible, orall active inhibitor of protein arginine deiminases (PADs) with IC50 of 0.8, 6.2, and 5.9 µM for PAD1, PAD3, and PAD4, respectively. |