GPR109A (Niacin Receptor 1) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofGPR109A (Niacin Receptor 1) GPR109A (Niacin Receptor 1)

Cat. No.	Product Name	Information
PC-21427	MK-1903 GPR109A agonist	MK-1903 is potent and selective agonist of GPR109a with EC50 of 12.9 nM, Emax 102%.
PC-43317	MK-0354 GPR109A agonist	MK-0354 is a potent, selective niacin receptor GPR109A partial agonist with EC50 of 1.65 and 1.08 uM for hGPR109A and mGPR109A in the whole cell cAMP assays.
PC-42694	MK-6892 GPR109A agonist	MK-6892 is a potent and selective high affinity niacin receptor (GPR109A) full agonist with Ki of 4.0 nM, EC50 of 16 nM in GTPγS assay.
PC-23376	HCAR3 agonist 5c HCAR3 agonist	HCAR3 agonist 5c (GPR109b agonist 5c) is a highly subtype-specific agonist of hydroxycarboxylic acid receptor 3 (HCAR3, GPR109B) with pEC50 of 7.53 and SPR KD of 47 nM, shows no activity against GPR109a.
PC-21439	GSK256073 GPR109A agonist	GSK256073 is a highly potent, selective agonist of hydroxy-carboxylic acid receptor 2 (HCA2, HM74A/GPR109A) with pEC50 of 7.5, 100-fold selective over HCA3 (pEC50=5.6).
PC-21426	SCH900271 GPR109A agonist	SCH900271 is a potent nicotinic acid receptor GPR109A agonist with EC50 of 2 nM in hu-GPR109a assays.

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