CGRP Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-42517	MK-3207 hydrochloride CGRP inhibitor	MK-3207 hydrochloride is a highly potent, selective CGRP receptor antagonist with Ki of 21 pM in in vitro binding assay and IC50 of 0.12 nM in cell-based functional assay.
PC-42516	MK-3207 CGRP antagonist	MK-3207 is a highly potent, selective CGRP receptor antagonist with Ki of 21 pM in in vitro binding assay and IC50 of 0.12 nM in cell-based functional assay.
PC-27352	PRT-064040 CGRP antagonist	PRT-064040 is a potent, selective calcitonin gene-related peptide receptor (CGRP) antagonist with binding Ki of 26.67 pM (human CGRP receptor), effectively inhibits human αCGRP-induced cAMP production with IC50 of 22.29 pM.
PC-24985	CGRP receptor antagonist 15 CGRP inhibitor	CGRP receptor antagonist 15 is a highly potent, orally bioavailable calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.029 nM and cAMP IC50 of 0.17 nM.

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