Cat. No. |
Product Name |
Information |
PC-23973 |
CCG258747
GRK2 inhibitor
|
CCG258747 is a potent selective GRK2 inhibitor with IC50 of 18 nM, 83-fold selectivity over GRK5. |
PC-23911 |
GRK5-IN-2
GRK5 inhibitor
|
GRK5-IN-2 (Compound 707)is a potent, selective G-protein-coupled receptor kinase 5 (GRK5) inhibitor with IC50 of 49.7 uM in luminescent ADP detection assay. |
PC-21461 |
GRL018-21
GRK5 inhibitor
|
GRL018-21 is a highly selective, potent, and non-covalent GRK5 inhibitor with IC50 of 10 nM, >100,000-fold selectivity over GRK2. |