| Cat. No. |
Product Name |
Information |
| PC-23974 |
CCG258208
GRK2 inhibitor
|
CCG258208 is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5. |
| PC-23973 |
CCG258747
GRK2 inhibitor
|
CCG258747 is a potent selective GRK2 inhibitor with IC50 of 18 nM, 83-fold selectivity over GRK5. |
| PC-21461 |
GRL018-21
GRK5 inhibitor
|
GRL018-21 is a highly selective, potent, and non-covalent GRK5 inhibitor with IC50 of 10 nM, >100,000-fold selectivity over GRK2. |