Diglyceride Acyltransferase (DGAT) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofDiglyceride Acyltransferase (DGAT) Diglyceride Acyltransferase (DGAT)

Cat. No.	Product Name	Information
PC-42121	A-922500 DGAT-1 inhibitor	A-922500 (A922500) is a potent, selective and orally bioavailable DGAT-1 inhibitor with IC50 of 9 and 22 nM against human and mouse DGAT-1, respectively.
PC-45795	T863 DGAT1 inhibitor	T-863 is a potent and selective, cell-permeable DGAT1 inhibitor that binds to the oleoyl-CoA binding pocket of DGAT1 with IC50 of 17 nM in TLC assay.
PC-21285	PF-07202954 DGAT2 inhibitor	PF-07202954 is a potent, selective next-generation DGAT2 inhibitor with IC50 of 10 nM (hDGAT2).
PC-21222	TP-020 MGAT2 inhibitor	TP-020 is a potent, selective, orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively.
PC-21221	BMS-986172 MGAT2 inhibitor	BMS-986172 is a highly potent, selective monoacylglycerol acyltransferase 2 (MGAT2) inhibitor with IC50 of 4.6 nM (human MGAT2).
PC-62952	JTT-553 benzosulfonate	JTT-553 is a novel potent, selective DGAT-1 inhibitor with IC50 of 2.38 nM, shows no inhibitory activity for human DGAT2 and ACA T1 (IC50>10 uM).

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