Neurotensin Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-60948	SR142948 Neurotensin receptor antagonist	SR142948 is a potent, selective and orally active neurotensin receptor antagonist with IC50 of 1.19 nM.
PC-60947	SR48692 NTSR1 antagonist	SR48692 (Meclinertant) is a potent, selective and orally active nonpeptide antagonist of neurotensin receptor NTSR1 with IC50 of 0.99 nM (guinea pig), without any intrinsic agonist activity.
PC-27369	NT150 NTSR2 agonist	NT150 (NT-150) is a potent, selective metabolically stable neurotensin receptor 2 (NTS2, NTSR2) agonist with Ki of 2.8 nM, has 22,000-fold selectivity over NTSR1.
PC-26998	Levocabastine hydrochloride NTSR2 antagonist	Levocabastine hydrochloride (R 50547) is a potent and selective histamine H1-receptor (H1R) antagonist, is also a selective, high affinity neurotensin receptor subtype 2 (NTSR2, NTS2) antagonist with Ki of 17 nM for mNTRS2.
PC-26997	NTRC-808 NTSR2 agonist	NTRC-808 is a potent, selective nonpeptide partial agonist of GPCR neurotensin receptor type 2 (NTS2, NTSR2) with EC50 of 14 nM and Ki of 88 nM, is selective for NTS2 versus NTS1.

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