Zavegepant (Vazegepant, BHV-3500) | CGRP antagonist | Probechem Biochemicals

Chemical Structure : Zavegepant

CAS No.: 1337918-83-8

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Zavegepant (Vazegepant, BHV-3500, BMS-742413)

货号: PC-38690Not For Human Use, Lab Use Only.

Zavegepant (Vazegepant, BHV-3500, BMS-742413) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.

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5 mg	￥1980	In stock
10 mg	￥2980	In stock
25 mg	￥4880	In stock
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100 mg		Get quote

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生物&药学活性

Zavegepant (Vazegepant, BHV-3500, BMS-742413) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.

物理化学性质&存储条件

分子量	638.817
分子式	C36H46N8O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)piperazin-1-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide

参考文献

1. Stephen E Mercer, et al. Bioorg Med Chem Lett. 2021 Jan 1;31:127624.

Zavegepant (Vazegepant, BHV-3500, BMS-742413)

生物&药学活性

物理化学性质&存储条件

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Zavegepant (Vazegepant, BHV-3500, BMS-742413)

生物&药学活性

物理化学性质&存储条件

参考文献

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