VU6077564 | mAChR M1 antagonist | Probechem Biochemicals

Chemical Structure : VU6077564

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VU6077564 (VU 6077564, VU-6077564)

货号: PC-27274Not For Human Use, Lab Use Only.

VU6077564 is a peripherally restricted and selective mAChR M1 antagonist with IC50 of 31 nM (hM1), >300-fold selective over hM2.

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生物&药学活性

VU6077564 is a peripherally restricted and selective mAChR M1 antagonist with IC50 of 31 nM (hM1), >300-fold selective over hM2.
VU6077564 exhibits potent KB value of 30 nM for human M1.
VU6077564 increases neurite outgrowth of adult rat sensory neurons with ED50 of 55 nM.

物理化学性质&存储条件

分子量	522.60
分子式	C26H27FN6O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-((1R,3s)-3-((S)-4-(5-Cyano-6-methylpyridin-2-yl)-2-methylpiperazine-1-carbonyl)cyclobutyl)-8-fluoroquinoline-5-sulfonamide

参考文献

1. Tomayo I Berida, et al. ACS Chem Neurosci. 2026 Jul 7. doi: 10.1021/acschemneuro.6c00367.

VU6077564 (VU 6077564, VU-6077564)

生物&药学活性

物理化学性质&存储条件

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VU6077564 (VU 6077564, VU-6077564)

生物&药学活性

物理化学性质&存储条件

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