VU6028418 | M4 mAChR antagonist | Probechem Biochemicals

Chemical Structure : VU6028418

CAS No.: 2649803-05-2

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货号: PC-72783Not For Human Use, Lab Use Only.

VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).

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VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).

分子量	432.491
分子式	C23H27F3N4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	rel-(3aR,6aS)-Octahydro-2-[(tetrahydro-2H-pyran-4-yl)methyl]-N-[6-(2,3,5-trifluorophenyl)-3-pyridazinyl]cyclopenta[c]pyrrol-5-amine

1. Matthew Spock, et al. ACS Med Chem Lett. 2021 Aug 2;12(8):1342-1349.