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首页-小分子抑制剂&激动剂-GPCR-mAChR-VU6015241
VU6015241

Chemical Structure : VU6015241

CAS No.: 2264025-00-3

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VU6015241 (VU 6015241)

货号: PC-72662Not For Human Use, Lab Use Only.

VU6015241 (VU 6015241) is a highly potent and selective antagonist of M4 muscarinic acetylcholine receptor (mAChR4) with IC50 of 71 nM.

规格 价格 库存 数量
2 mg ￥2980 In stock
5 mg ￥4980 In stock
10 mg ￥7880 In stock
25 mg Get quote
100 mg Get quote
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纯度 & COA & 质检文件 纯度: 99.53% (HPLC) Select Batch:

生物&药学活性

VU6015241 (VU 6015241) is a highly potent and selective antagonist of M4 muscarinic acetylcholine receptor (mAChR4) with IC50 of 71 nM.
VU6015241 demonstrates selectivity across multiple species, excellent aqueous solubility, and moderate brain exposure in rodents after intraperitoneal administration.

物理化学性质&存储条件

分子量 449.599
分子式 C26H35N5O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-N-(4-(6-(((6-((tetrahydro-2H-pyran-4-yl)methyl)-6-azaspiro[2.5]octan-1-yl)methyl)amino)pyridazin-3-yl)phenyl)acetamide

参考文献

1. Aaron M Bender, et al. Bioorg Med Chem Lett. 2022 Jan 15;56:128479.

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