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首页-小分子抑制剂&激动剂-GPCR-mAChR-VU0415248
VU0415248

Chemical Structure : VU0415248

CAS No.: 1359087-83-4

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VU0415248 (VU 0415248)

货号: PC-20508Not For Human Use, Lab Use Only.

VU0415248 is a highly selective antagonist of muscarinic acetylcholine receptor subtype 1 (M1 mAChR) with IC50 of 0.4 uM and 0.18 uM for hM1R and rM1R, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

VU0415248 is a highly selective antagonist of muscarinic acetylcholine receptor subtype 1 (M1 mAChR) with IC50 of 0.4 uM and 0.18 uM for hM1R and rM1R, respectively.
VU0415248 shows very high selectivity for the M1 receptor over the M2–5 subtypes across all five human and rat receptors.

物理化学性质&存储条件

分子量 425.51
分子式 C21H23N5O3S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

O=S(C1=CC=CC2=C1C=CC=N2)(NCCC(N3CCN(C4=CC=NC=C4)CC3)=O)=O

参考文献

1. Bruce J Melancon, et al. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1044-8.

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