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首页-小分子抑制剂&激动剂-GPCR-Lysophospholipid Receptor-TY-52156
TY-52156

Chemical Structure : TY-52156

CAS No.: 934369-14-9

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TY-52156 (TY52156)

货号: PC-21209Not For Human Use, Lab Use Only.

TY-52156 is a potent, selective S1P3 receptor antagonist with Ki of 110 nM.

规格 价格 库存 数量
25 mg ￥1980 In stock
50 mg ￥2980 In stock
100 mg ￥4880 In stock
1 g Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

TY-52156 is a potent, selective S1P3 receptor antagonist with Ki of 110 nM.
TY-52156 preferentially inhibited the S1P-induced increase in [Ca2]i in S1P3-CHO rather than S1P1-, S1P2-CHO, and S1P4-Chem.
TY-52156 inhibited both the S1P-induced increase in [Ca(2+)](i) and Rho activation in human coronary artery smooth muscle cells.
TY-52156 inhibited FTY-720-induced S1P(3) receptor-mediated bradycardia in vivo.

物理化学性质&存储条件

分子量 364.27
分子式 C18H19Cl2N3O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-(4-chlorophenylhydrazono)-1-(4-chlorophenylamino)-3,3-dimethyl- 2-butanone

参考文献

1. Murakami A, et al. Mol Pharmacol. 2010 Apr;77(4):704-13.

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