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首页-小分子抑制剂&激动剂-GPCR-Lysophospholipid Receptor-TP0541640
TP0541640

Chemical Structure : TP0541640

CAS No.: 2604363-47-3

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TP0541640 (TP 0541640)

货号: PC-21122Not For Human Use, Lab Use Only.

TP0541640 (TP 0541640) is a novel potent LPA1 antagonist with IC50 of 1.6 nM, shows potential for the treatment of lung and skin fibrosis.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    TP0541640 (TP 0541640) is a novel potent LPA1 antagonist with IC50 of 1.6 nM, shows potential for the treatment of lung and skin fibrosis.
    TP0541640 (10, 30, or 100 mg/kg) suppressed LPA-induced histamine release in C57BL6 mice.
    TP0541640 shows anti-fibrotic effects suppressive effect in mouse model of bleomycin-induced skin fibrosis.

    物理化学性质&存储条件

    分子量 504.57
    分子式 C27H34F2N2O5
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    1-({[(1 R)-1-(3,5-dimethoxy-4-methylphenyl)ethyl](4-phenylbutyl)carbamoyl}amino)-3,3-difluorocyclobutane-1-carboxylic acid

    参考文献

    1. Yuki Kobayashi, et al. Eur J Med Chem. 2023 Aug 20;260:115749.

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