THRX-198321 |CAS:743460-20-0 Probechem Biochemicals

Chemical Structure : THRX-198321

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THRX-198321 (THRX198321)

货号: PC-63038Not For Human Use, Lab Use Only.

THRX-198321 is a bifunctional mAChR antagonist and β2-adrenoceptor agonist (MABA) with pKi of 9.69/10.05 for M1/M2 respectively, pEC50 of 9.25 for β2AR.

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生物&药学活性

THRX-198321 is a bifunctional mAChR antagonist and β2-adrenoceptor agonist (MABA) with pKi of 9.69/10.05 for M1/M2 respectively, pEC50 of 9.25 for β2AR.
THRX-198321 exhibits a multivalent bimodal orientation in the orthosteric and allosteric binding pockets of mAChR and β(2)AR.

物理化学性质&存储条件

分子量	640.825
分子式	C38H48N4O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Biphenyl-2-yl-carbamic acid 1-{9-[(R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydro-quinolin-5-yl)-ethylamino]-nonyl}-piperidin-4-yl ester

参考文献

1. Steinfeld T, et al. Mol Pharmacol. 2011 Mar;79(3):389-99.

THRX-198321 (THRX198321)

生物&药学活性

物理化学性质&存储条件

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THRX-198321 (THRX198321)

生物&药学活性

物理化学性质&存储条件

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