TDO2 inhibitor Cpd-1

Chemical Structure : TDO2 inhibitor Cpd-1

加入收藏

货号: PC-23417Not For Human Use, Lab Use Only.

TDO2 inhibitor Cpd-1 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 327 nM in human TDO2 cellular assay utilizing SW48 cells.

规格	价格	库存	数量
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

TDO2 inhibitor Cpd-1 is a potent, selective small molecule inhibitor of the apo form of human TDO2 with IC50 of 327 nM in human TDO2 cellular assay utilizing SW48 cells.
TDO2 inhibitor Cpd-1 showed almost no inhibition of IDO1, with respective IC50 values of 5.7 µM.

物理化学性质&存储条件

分子量	532.64
分子式	C30H36N4O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl 9-(3-(2-propylphenyl)-1-(1-phenylethyl)ureido)-2-methoxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-3-carboxylate

参考文献

1. Lotz-Jenne C, et al. Sci Rep. 2024 Nov 14;14(1):27937.