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首页-小分子抑制剂&激动剂-Wnt/Notch/Hedgehog-Casein Kinase-SR-2890
SR-2890

Chemical Structure : SR-2890

CAS No.: 1454584-91-8

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SR-2890 (SR 2890, SR2890)

货号: PC-60580Not For Human Use, Lab Use Only.

SR-2890 is a potent, highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitor with IC50 of 4 nM for CK1δ.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    SR-2890 is a potent, highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitor with IC50 of 4 nM for CK1δ.
    SR-2890 inhibits melanoma A375 cell growth with EC50 of 38 nM in MTT assays.
    SR-2890 has physical, in vitro and in vivo PK properties suitable for use in proof of principle animal xenograft studies against human cancer cell lines.

    物理化学性质&存储条件

    分子量 477.932
    分子式 C23H21ClFN9
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-((5-chloro-1H-benzo[d]imidazol-2-yl)methyl)-9-(3-fluorophenyl)-2-(piperazin-1-yl)-9H-purin-6-amine

    参考文献

    1. Bibian M, et al. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4374-80.

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