SAR-100842 |CAS:1195941-38-8 Probechem Biochemicals

Chemical Structure : SAR-100842

CAS No.: 1195941-38-8

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SAR-100842 (Fipaxalparant, SAR100842)

货号: PC-35275Not For Human Use, Lab Use Only.

Fipaxalparant (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays.

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5 mg	￥2480	In stock
10 mg	￥3980	In stock
25 mg	￥5980	In stock
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100 mg		Get quote

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生物&药学活性

Fipaxalparant (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays.
Fipaxalparant (SAR100842) demonstrates potential for the treatment of systemic sclerosis and related fibrotic diseases.

物理化学性质&存储条件

分子量	445.515
分子式	C27H27NO5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-{4-methoxy-3-[2-(3-methylphenyl)ethoxy]benzamido}-2,3-dihydro-1H-indene-2-carboxylic acid

参考文献

1. Ellery J, et al. Eur J Pharmacol. 2018 May 26;833:8-15.

2. Kihara Y, et al. Exp Cell Res. 2015 May 1;333(2):171-7.

SAR-100842 (Fipaxalparant, SAR100842)

生物&药学活性

物理化学性质&存储条件

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SAR-100842 (Fipaxalparant, SAR100842)

生物&药学活性

物理化学性质&存储条件

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