Pitolisant oxalate | H3 receptor antagonist | Probechem Biochemicals

Chemical Structure : Pitolisant oxalate

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Pitolisant oxalate (Tiprolisant oxalate)

货号: PC-42910Not For Human Use, Lab Use Only.

Pitolisant oxalate (Tiprolisant oxalate) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

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生物&药学活性

Pitolisant oxalate (Tiprolisant oxalate) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
Pitolisant oxalate has no effect on H1, H2, H4 receptors (IC50>10 uM); orally bioactive.

物理化学性质&存储条件

分子量	385.8823
分子式	C19H28ClNO5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-, ethanedioate (1:1)

参考文献

1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.

2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.

3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.

Pitolisant oxalate (Tiprolisant oxalate)

生物&药学活性

物理化学性质&存储条件

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Pitolisant oxalate (Tiprolisant oxalate)

生物&药学活性

物理化学性质&存储条件

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