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首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-Pitolisant
Pitolisant

Chemical Structure : Pitolisant

CAS No.: 362665-56-3

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Pitolisant (Tiprolisant, BF-2649, BF 2.649)

货号: PC-42909Not For Human Use, Lab Use Only.

Pitolisant (Tiprolisant, BF-2649, BF 2.649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

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10 mg ￥780 In stock
25 mg ￥1380 In stock
50 mg ￥2180 In stock
100 mg ￥3580 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Pitolisant (Tiprolisant, BF-2649, BF 2.649) is a potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
Pitolisant shows no effect on H1, H2, H4 receptors (IC50>10 uM).
Pitolisant is orally bioactive.

物理化学性质&存储条件

分子量 295.8474
分子式 C17H26ClNO
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-

参考文献

1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.

2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.

3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.

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