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首页-小分子抑制剂&激动剂-GPCR-Lysophospholipid Receptor-ONO-7300243
ONO-7300243

Chemical Structure : ONO-7300243

CAS No.: 638132-34-0

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ONO-7300243 (ONO7300243;ONO 7300243)

货号: PC-42284Not For Human Use, Lab Use Only.

ONO7300243 is a novel potent, selective, orally available lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 uM.

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25 mg ￥2180 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

ONO7300243 is a novel potent, selective, orally available lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 uM.
ONO7300243 exhibits good selectivity (>50-fold) toward LPA1over LPA2; shows good efficacy in vivo, reduces intraurethral pressure in rats without affecting the blood pressure (30mg/kg. p.o.).

物理化学性质&存储条件

分子量 461.54944
分子式 C28H31NO5
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Benzeneacetic acid, 4-[[(3,5-dimethoxy-4-methylbenzoyl)(3-phenylpropyl)amino]methyl]-

参考文献

1. Terakado M, et al. ACS Med Chem Lett. 2016 Aug 19;7(10):913-918.

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