Mirabegron | β3-adrenoceptor agonist | Probechem Biochemicals

Chemical Structure : Mirabegron

CAS No.: 223673-61-8

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Mirabegron (YM178, YM-178)

货号: PC-21196Not For Human Use, Lab Use Only.

Mirabegron (YM178) is a potent, selective selective β3-adrenoceptor agonist with EC50 of 22.4 nM.

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25 mg	￥2280	In stock
50 mg	￥3980	In stock
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1 g		Get quote

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生物&药学活性

Mirabegron (YM178) is a potent, selective selective β3-adrenoceptor agonist with EC50 of 22.4 nM.
Mirabegron (YM178) displays no activity against human beta1- and beta2-ARs.
Mirabegron (YM178) exhibited relaxant effects of YM178 were evaluated in rats and humans bladder strips precontracted with carbachol (CCh.
Mirabegron (YM178) (3 mg/kg, i.v.) decreased the frequency of rhythmic bladder contraction induced by intravesical filling with saline without suppressing its amplitude in anesthetized rats.

物理化学性质&存储条件

分子量	396.51
分子式	C21H24N4O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-2-(2-aminothiazol-4-yl)-4'-{2-[(2-hydroxy-2-phenylethyl)amino]-ethyl} acetanilide

参考文献

1. Takasu T, et al. J Pharmacol Exp Ther. 2007 May;321(2):642-7.

Mirabegron (YM178, YM-178)

生物&药学活性

物理化学性质&存储条件

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Mirabegron (YM178, YM-178)

生物&药学活性

物理化学性质&存储条件

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