LSN3172176 |CAS: 3033820-85-5 Probechem Biochemicals

Chemical Structure : LSN3172176

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LSN3172176 (LSN-3172176)

货号: PC-63443Not For Human Use, Lab Use Only.

LSN3172176 is a potent, selectiive M1 mAChR partial agonist (EC50 2.4-7.0nM, Emax 43%-73%), shows binding selectivity for M1 mAChRs (Kd=1.5 nM).

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生物&药学活性

LSN3172176 is a potent, selectiive M1 mAChR partial agonist (EC50 2.4-7.0nM, Emax 43%-73%), shows binding selectivity for M1 mAChRs (Kd=1.5 nM).
LSN3172176 is a potential PET tracer for assessment of M1 mAChR target engagement in the clinic and to further elucidate the function of M1 mAChRs in health and disease.

物理化学性质&存储条件

分子量	385.508
分子式	C22H31N3O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl 4-(6-methyl-2-oxoindolin-1-yl)-[1,4'-bipiperidine]-1'-carboxylate

参考文献

1. Mogg AJ, et al. J Pharmacol Exp Ther. 2018 Apr 11. pii: jpet.117.246454.

LSN3172176 (LSN-3172176)

生物&药学活性

物理化学性质&存储条件

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LSN3172176 (LSN-3172176)

生物&药学活性

物理化学性质&存储条件

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