LPA2 antagonist 1 |CAS:1017606-66-4 Probechem Biochemicals

Chemical Structure : LPA2 antagonist 1

CAS No.: 1017606-66-4

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LPA2 antagonist 1 (LPA2-IN-1)

货号: PC-45411Not For Human Use, Lab Use Only.

LPA2 antagonist 1 is a potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM.

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10 mg	￥4580	In stock
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生物&药学活性

LPA2 antagonist 1 is a potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM.
LPA2 antagonist 1 inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner.
LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner.

物理化学性质&存储条件

分子量	500.4649
分子式	C20H23Cl2N5O2S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Thieno[3,2-d]pyrimidin-4-amine, N-[(1S)-2-[4-[(3,4-dichlorophenyl)sulfonyl]-1-piperazinyl]-1-methylethyl]-7-methyl-

参考文献

1. Beck HP, et al. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.

LPA2 antagonist 1 (LPA2-IN-1)

生物&药学活性

物理化学性质&存储条件

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LPA2 antagonist 1 (LPA2-IN-1)

生物&药学活性

物理化学性质&存储条件

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