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首页-小分子抑制剂&激动剂-GPCR-Histamine Receptor-LINS01022
LINS01022

Chemical Structure : LINS01022

CAS No.: 2757222-80-1

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LINS01022 (LINS-01022)

货号: PC-27866Not For Human Use, Lab Use Only.

LINS01022 is a high affinity, selective histamine H3 receptor (H3R) antagonist with pKi of 8.2, >1000-fold selective over H4R, exhibits potent antiproliferative effect against 4T1 and MDA-MB-231 TNBC cell lines.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

LINS01022 is a high affinity, selective histamine H3 receptor (H3R) antagonist with pKi of 8.2, >1000-fold selective over H4R, exhibits potent antiproliferative effect against 4T1 and MDA-MB-231 TNBC cell lines.

物理化学性质&存储条件

分子量 288.39
分子式 C17H24N2O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-allyl-4-((5-methoxy-2,3-dihydrobenzofuran-2-yl)methyl)piperazine

参考文献

1. Lopes FB, et al. Chem Biol Drug Des. 2022 Nov;100(5):722-729.

2. Ospital IA, et al. Biomed Pharmacother. 2024 May;174:116527.

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