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首页-小分子抑制剂&激动剂-GPCR-Lysophospholipid Receptor-H2L5186303
H2L5186303

Chemical Structure : H2L5186303

CAS No.: 139262-76-3

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H2L5186303 (H2L 5186303)

货号: PC-49229Not For Human Use, Lab Use Only.

H2L5186303 is a potent, selective LPA2 receptor antagonist with IC50 of 8.9 nM, no significant activity against LPA1 and LPA3 receptors (IC50>1,000 nM), inhibits LPA(2) mediated Erk activation and proliferation of HCT-116 cells.

规格 价格 库存 数量
5 mg ￥1380 In stock
10 mg ￥2180 In stock
25 mg ￥3780 In stock
50 mg ￥5880 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

H2L5186303 is a potent, selective LPA2 receptor antagonist with IC50 of 8.9 nM, no significant activity against LPA1 and LPA3 receptors (IC50>1,000 nM), inhibits LPA(2) mediated Erk activation and proliferation of HCT-116 cells.

物理化学性质&存储条件

分子量 488.452
分子式 C26H20N2O8
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Butenoic acid, 4,4′-[1,3-phenylenebis(oxy-4,1-phenyleneimino)]bis[4-oxo-, (Z,Z)-

参考文献

1. Hilary P Beck, et al. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.

2. Chabowski DS, et al. Br J Pharmacol. 2018 Nov;175(22):4266-4280.

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