GD136 (VUF10775) | H1R/H4R antagonist | Probechem Biochemicals

Chemical Structure : GD136

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GD136 (GD-136, VUF10775, VUF-10775)

货号: PC-28138Not For Human Use, Lab Use Only.

GD136 (GD-136) is a potent, selective dual histamine H1 and H4 receptors (H1R/H4R) ligand / antagonist with pKi of 7.61 and 7.93 (hH1R/hH4R), shows >100-fold selectivity over hH2R and hH3R.

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生物&药学活性

GD136 (VUF10775, GD-136) is a potent, selective dual histamine H1 and H4 receptors (H1R/H4R) ligand / antagonist with pKi of 7.61 and 7.93 (hH1R/hH4R), shows >100-fold selectivity over hH2R and hH3R.

物理化学性质&存储条件

分子量	494.54
分子式	C22H25F3N6O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)quinazolin-4-yl)amino)-N-phenylethane-1-sulfonamide

参考文献

1. Weber P, et al. J Med Chem. 2026 Sep 10;69(17):20967-21003.

GD136 (GD-136, VUF10775, VUF-10775)

生物&药学活性

物理化学性质&存储条件

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GD136 (GD-136, VUF10775, VUF-10775)

生物&药学活性

物理化学性质&存储条件

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