Fesoterodine fumarate (PF-00695838) | mAChR antagonist

Chemical Structure : Fesoterodine fumarate

CAS No.: 286930-03-8

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Fesoterodine fumarate (PF-00695838 fumarate, SPM907, SPM-907)

货号: PC-61893Not For Human Use, Lab Use Only.

Fesoterodine fumarate (PF-00695838) is a competitive muscarinic receptor antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors.

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生物&药学活性

Fesoterodine fumarate (PF-00695838) is a competitive muscarinic receptor antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors.
Fesoterodine has muscle relaxant and urinary antispasmodic properties.
Fesoterodine binds and inhibits muscarinic receptors on the bladder detrusor muscle, prevents bladder contractions or spasms caused by acetylcholine.

物理化学性质&存储条件

分子量	527.658
分子式	C30H41NO7
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	[2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-(hydroxymethyl)phenyl] 2-methylpropanoate fumarate

参考文献

1. Ney P, et al. BJU Int. 2008 Apr;101(8):1036-42.

2. Michel MC. Expert Opin Pharmacother. 2008 Jul;9(10):1787-96.

3. Chapple CR, et al. BJU Int. 2008 Nov;102(9):1128-32.

Fesoterodine fumarate (PF-00695838 fumarate, SPM907, SPM-907)

生物&药学活性

物理化学性质&存储条件

参考文献

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Fesoterodine fumarate (PF-00695838 fumarate, SPM907, SPM-907)

生物&药学活性

物理化学性质&存储条件

参考文献

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