DREADD agonist compound 21 | hM3Dq agonist | Probechem Biochemicals

Chemical Structure : DREADD agonist compound 21

CAS No.: 56296-18-5

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DREADD agonist compound 21 (DREADD agonist 21, hM3Dq agonist)

货号: PC-42096Not For Human Use, Lab Use Only.

DREADD agonist compound 21 (hM3Dq agonist) is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.

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10 mg	￥1480	In stock
25 mg	￥2580	In stock
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生物&药学活性

DREADD agonist compound 21 (hM3Dq agonist) is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.
hM3Dq-agonist-21 displays 3.5-fold selective over H1, 40-fold selective over 5HT2A, 100-fold selective over 5HT2C, 165-fold selective over α1A, and inactive at native human M3 receptor (hM3).

物理化学性质&存储条件

分子量	278.3516
分子式	C17H18N4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 78 mg/mL
Chemical Name/SMILES	5H-Dibenzo[b,e][1,4]diazepine, 11-(1-piperazinyl)-

参考文献

1. Chen X, et al. ACS Chem Neurosci. 2015 Mar 18;6(3):476-84.

DREADD agonist compound 21 (DREADD agonist 21, hM3Dq agonist)

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DREADD agonist compound 21 (DREADD agonist 21, hM3Dq agonist)

生物&药学活性

物理化学性质&存储条件

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