DKR-1051 |CAS:2089053-14-3 Probechem Biochemicals

Chemical Structure : DKR-1051

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DKR-1051 (DKR 1051;DKR1051)

货号: PC-61102Not For Human Use, Lab Use Only.

DKR-1051 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 61 nM, 9-fold selectivity over sigma 1 receptors (Ki=556 nM).

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生物&药学活性

DKR-1051 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 61 nM, 9-fold selectivity over sigma 1 receptors (Ki=556 nM).
DKR-1051 modulates intracellular Ca2+ levels in human SK-N-SH neuroblastoma cells。
DKR-1051 relieves spared nerve injury-induced mechanical hypersensitivity in vivo.

物理化学性质&存储条件

分子量	385.474
分子式	C24H26F3N
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,6R)-2-cyclopentyl-9-(4-(trifluoromethyl)phenyl)-1,2,3,4,5,6-hexahydro-1,6-methanobenzo[c]azocine

参考文献

1. Yi B, et al. J Neurochem. 2017 Feb;140(4):561-575.

2. Sahn JJ, et al. ACS Chem Neurosci. 2017 Aug 16;8(8):1801-1811.

DKR-1051 (DKR 1051;DKR1051)

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DKR-1051 (DKR 1051;DKR1051)

生物&药学活性

物理化学性质&存储条件

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