Clobenpropit (VUF-9153) | Histamine H3 antagonist | Probechem Biochemicals

Chemical Structure : Clobenpropit

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Clobenpropit (VUF-9153, VUF9153)

货号: PC-35222Not For Human Use, Lab Use Only.

Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.

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生物&药学活性

Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.
Clobenpropit (VUF-9153) increases brain histidine decarboxylase activity dose dependently, inhibits electrically induced convulsions in mice.

物理化学性质&存储条件

分子量	308.828
分子式	C14H17ClN4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Carbamimidothioic acid, [(4-chlorophenyl)methyl]-, 3-(1H-imidazol-4-yl)propyl ester (9CI)

参考文献

1. Yokoyama H, et al. Eur J Pharmacol. 1994 Jul 21;260(1):23-8.

2. Clark EA, et al. Br J Pharmacol. 1995 Jan;114(2):357-62.

3. Stark H, et al. J Med Chem. 1996 Mar 1;39(5):1157-63.

4. Mochizuki T, et al. Brain Res. 1996 Dec 16;743(1-2):178-83.

Clobenpropit (VUF-9153, VUF9153)

生物&药学活性

物理化学性质&存储条件

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Clobenpropit (VUF-9153, VUF9153)

生物&药学活性

物理化学性质&存储条件

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