CL 316243 disodium |CAS:138908-40-4 Probechem Biochemicals

Chemical Structure : CL 316243 disodium

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CL 316243 disodium (CL316243 disodium)

货号: PC-62016Not For Human Use, Lab Use Only.

CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.

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生物&药学活性

CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
CL 316243 displays >10000-fold selective over β1 and β2 receptors。
CL 316243 significantly increases brown adipose tissue thermogenesis and resting metabolic rate in mice, also increases the concentration of insulin receptors and decreases the levels of serum insulin and blood glucose during the glucose overloading test.

物理化学性质&存储条件

分子量	465.8
分子式	C20H18ClNNa2O7
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-[(2R)-2-[[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino]propyl]-1,3-benzodioxole-2,2-dicarboxylic acid disodium salt

参考文献

1. Berlan M, et al. J Pharmacol Exp Ther. 1994 Mar;268(3):1444-51.

2. Himms-Hagen J, et al. Am J Physiol. 1994 Apr;266(4 Pt 2):R1371-82.

3. Yoshida T, et al. Life Sci. 1994;54(7):491-8.

CL 316243 disodium (CL316243 disodium)

生物&药学活性

物理化学性质&存储条件

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CL 316243 disodium (CL316243 disodium)

生物&药学活性

物理化学性质&存储条件

参考文献

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