CAM4066 | CK2α inhibitor | Probechem Biochemicals

Chemical Structure : CAM4066

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CAM4066 (CAM 4066, CAM-4066)

货号: PC-35184Not For Human Use, Lab Use Only.

CAM4066 (CAM-4066) is a potent and selective CK2alpha (CK2α) inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.

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生物&药学活性

CAM4066 (CAM-4066) is a potent and selective CK2alpha (CK2α) inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.
CAM4066 inhibits CK2 activity by exploiting a pocket located outside the ATP binding site (alphaD pocket).

物理化学性质&存储条件

分子量	479.961
分子式	C26H26ClN3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(3-(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)propanamido)propanamido)benzoic acid

参考文献

1. Iegre J, et al. Chem Sci. 2018 Feb 20;9(11):3041-3049.

2. Brear P, et al. Chem Sci. 2016 Nov 1;7(11):6839-6845.

3. De Fusco C, et al. Bioorg Med Chem. 2017 Jul 1;25(13):3471-3482.

CAM4066 (CAM 4066, CAM-4066)

生物&药学活性

物理化学性质&存储条件

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CAM4066 (CAM 4066, CAM-4066)

生物&药学活性

物理化学性质&存储条件

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