BAY-6096 | Adrenergic α2B inhibitor | Probechem Biochemicals

Chemical Structure : BAY-6096

加入收藏

BAY-6096 (BAY6096)

货号: PC-20307Not For Human Use, Lab Use Only.

BAY-6096 (BAY6096) is a potent, selective, and highly water-soluble adrenergic α2B antagonist with IC50 of 14 nM.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

BAY-6096 (BAY6096) is a potent, selective, and highly water-soluble adrenergic α2B antagonist with IC50 of 14 nM.
BAY-6096 displays >350-fold selectivity over α1A, α2A and α2C.
BAY-6096 shows high water-solublity (90 mg/mL), could be formulated in 0.9% NaCl solution showed no adsorption toward sterile filters and no instabilities upon heat steam sterilization.
BAY-6096 dose-dependently reduced blood pressure increases in rats induced by an α2B agonist.

物理化学性质&存储条件

分子量	426.91
分子式	C21H23ClN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-[2-({[3-(3,5-Dimethyl-1,2-oxazol-4-yl)imidazo[1,2-a]pyridin-7-yl]carbonyl}amino)ethyl]-4-(methylamino)pyridinium Chloride

参考文献

1. Daniel Meibom, et al. J Med Chem. 2023 Mar 18. doi: 10.1021/acs.jmedchem.2c01690.

BAY-6096 (BAY6096)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

BAY-6096 (BAY6096)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.