ASP8302 | M3 PAM | Probechem Biochemicals

Chemical Structure : ASP8302

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ASP8302 (ASP-8302, ASP 8302)

货号: PC-72280Not For Human Use, Lab Use Only.

ASP8302 (ASP 8302) is a potent, selective, positive allosteric modulator (PAM) of muscarinic M3 receptor.

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生物&药学活性

ASP8302 (ASP 8302) is a potent, selective, positive allosteric modulator (PAM) of muscarinic M3 receptor.
Threonine 230 (Thr 230) is the amino acid essential for the PAM effect of ASP8302.

物理化学性质&存储条件

分子量	590.158
分子式	C26H32ClN7O3S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-[(2S)-4-(5-{[4-(4-chlorothiophen-2-yl)-5-{[(2R)-2-methylpyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl]carbamoyl}pyrazin-2-yl)-2-methylpiperazin-1-yl]propanoic acid

参考文献

1. Okimoto R, et al. J Pharmacol Exp Ther. 2021 Oct;379(1):64-73.

2. Okimoto R, et al. Low Urin Tract Symptoms. 2022 Feb 12.

ASP8302 (ASP-8302, ASP 8302)

生物&药学活性

物理化学性质&存储条件

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ASP8302 (ASP-8302, ASP 8302)

生物&药学活性

物理化学性质&存储条件

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