ARV-766 | AR PROTAC | Probechem Biochemicals

Chemical Structure : ARV-766

CAS No.: 2750830-09-0

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ARV-766 (Luxdegalutamide, ARV766, ARV 766)

货号: PC-20665Not For Human Use, Lab Use Only.

ARV-776 (Luxdegalutamide, ARV776) is potent, orally bioavailable PROTAC androgen receptor (AR) degrader that degrades not only wild-type AR but also clinically relevant AR LBD mutants, including the most prevalent AR L702H, H875Y, and T878A mutations.

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5 mg	￥4580	In stock
10 mg	￥7280	In stock
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生物&药学活性

ARV-776 (Luxdegalutamide, ARV776) is potent, orally bioavailable PROTAC androgen receptor (AR) degrader that degrades not only wild-type AR but also clinically relevant AR LBD mutants, including the most prevalent AR L702H, H875Y, and T878A mutations.

物理化学性质&存储条件

分子量	807.97
分子式	C45H54FN7O6
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(4-((1-(4-(((1r,3r)-3-(4-cyano-3-methoxyphenoxy)-2,2,4,4-tetramethylcyclobutyl)carbamoyl)phenyl)piperidin-4-yl)methyl)piperazin-1-yl)-N-((S)-2,6-dioxopiperidin-3-yl)-2-fluorobenzamide

参考文献

1. Daniel P. Petrylak, et al. 2023 ASCO Genitourinary Cancers Symposium

ARV-766 (Luxdegalutamide, ARV766, ARV 766)

生物&药学活性

物理化学性质&存储条件

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ARV-766 (Luxdegalutamide, ARV766, ARV 766)

生物&药学活性

物理化学性质&存储条件

参考文献

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