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首页-小分子抑制剂&激动剂-GPCR-Lysophospholipid Receptor-ACT-1016-0707
ACT-1016-0707

Chemical Structure : ACT-1016-0707

CAS No.: 2569467-78-1

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ACT-1016-0707

货号: PC-21751Not For Human Use, Lab Use Only.

ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.
    ACT-1016-0707 suppressed the LPA-induced vascular leakage at a p.o. dose of 30 mg/kg.

    物理化学性质&存储条件

    分子量 438.93
    分子式 C19H23ClN4O4S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-(6-Chloro-4-methoxypyridin-3-yl)-3-(2-isopropylphenyl)-1-sulfamoylazetidine-3-carboxamide

    参考文献

    1. Lescop C, et al. J Med Chem. 2024 Feb 13. doi: 10.1021/acs.jmedchem.3c01827.

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