欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-nor-Binaltorphimine
nor-Binaltorphimine

Chemical Structure : nor-Binaltorphimine

CAS No.: 105618-26-6

加入收藏

nor-Binaltorphimine (Nor-BNI, Norbinaltorphimine)

货号: PC-27172Not For Human Use, Lab Use Only.

nor-Binaltorphimine (Nor-BNI, Norbinaltorphimine) is a potent, selective, long-acting competitive κ-opioid receptor (KOR) antagonist, blocks KOR-mediated analgesic effects, and inhibits butorphanol-induced changes in κ-opioid receptor binding kinetics, desensitization and down-regulation.

规格 价格 库存 数量
5 mg ￥1780 In stock
10 mg ￥2780 In stock
50 mg Get quote
100 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

nor-Binaltorphimine (Nor-BNI, Norbinaltorphimine) is a potent, selective, long-acting competitive κ-opioid receptor (KOR) antagonist, blocks KOR-mediated analgesic effects, and inhibits butorphanol-induced changes in κ-opioid receptor binding kinetics, desensitization and down-regulation.

物理化学性质&存储条件

分子量 661.80
分子式 C40H43N3O6
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(4bS,8R,8aS,10aS,11R,14aS,19aR,20bR)-7,12-bis(cyclopropylmethyl)-5,6,7,8,9,10,11,12,13,14,19a,20b-dodecahydro-20H-4,8:11,15-dimethanobis(benzofuro)[2,3-a:3',2'-i]dipyrido[4,3-b:3',4'-h]carbazole-1,8a,10a,18-tetraol

参考文献

1. Spanagel R, et al. Eur J Pharmacol. 1994;264(2):157-162.

2. Jaw SP, et al. Eur J Pharmacol. 1993;239(1-3):133-140.

备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

联系我们 sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

询单

  • *产品名称:
  • *姓名:
  • *邮箱:
  • *公司名称:
  • *询单数量:
  • *国籍:
  • 询单信息: