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首页-小分子抑制剂&激动剂-Immunology/Inflammation-PGE synthase-mPGES1-IN-16
mPGES1-IN-16

Chemical Structure : mPGES1-IN-16

CAS No.: 1915003-93-8

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mPGES1-IN-16

货号: PC-62820Not For Human Use, Lab Use Only.

mPGES1-IN-16 is a potent and selective mPGES-1 inhibitor with IC50 of 1 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    mPGES1-IN-16 is a potent and selective mPGES-1 inhibitor with IC50 of 1 nM.
    mPGES1-IN-16 displays no activity against a panel of 35 receptors, ion channels, and hERG.
    mPGES1-IN-16 shows IC50/IC80 of 6 nM/24 nM for inhibition of PGE2 formation in vitro in LPS-stimulated human whole blood (HWB); orally bioavailable in vivo.

    物理化学性质&存储条件

    分子量 485.628
    分子式 C30H35N3O3
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    2-(2-((1S,2S)-2-(1-(8-methylquinolin-2-yl)piperidine-4-carboxamido)cyclopentyl)ethyl)benzoic acid

    参考文献

    1. Partridge KM, et al. Bioorg Med Chem Lett. 2017 Mar 15;27(6):1478-1483.

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