Ziprasidone hydrochloride monohydrate | D2/5-HT2A antagonist

Chemical Structure : Ziprasidone hydrochloride monohydrate

CAS No.: 138982-67-9

加入收藏

Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate)

货号: PC-45229Not For Human Use, Lab Use Only.

Ziprasidone hydrochloride monohydrate (CP-88059) is a full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively.

规格	价格	库存
25 mg	￥880	In stock
50 mg	￥1380	In stock
100 mg	￥2180	In stock
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

Ziprasidone hydrochloride monohydrate (CP-88059) is a full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively.
Ziprasidone also is a partial agonist of 5-HT1A, and a partial antagonist of 5-HT2C and 5-HT1D receptors.
Ziprasidone exhibits potent antipsychotic activity in vivo.

物理化学性质&存储条件

分子量	467.4119
分子式	C21H24Cl2N4O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2H-Indol-2-one, 5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-, hydrochloride, hydrate (1:1:1)

参考文献

1. Mattei C, et al. J Cent Nerv Syst Dis. 2011 Feb 15;3:1-16.

2. Seeger TF, et al. J Pharmacol Exp Ther. 1995 Oct;275(1):101-13.

3. Schotte A, et al. Psychopharmacology (Berl). 1996 Mar;124(1-2):57-73.

Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.