Zatebradine |CAS:85175-67-3 Probechem Biochemicals

Chemical Structure : Zatebradine

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Zatebradine (UL-FS49)

货号: PC-43527Not For Human Use, Lab Use Only.

Zatebradine (UL-FS49) is a potent blocker (antagonist) of hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, a specific bradycardic agent.

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生物&药学活性

Zatebradine (UL-FS49) is a potent blocker (antagonist) of hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, a specific bradycardic agent.
Zatebradine (UL-FS49) blocks cardiac pacemaker current (If), decreases the rate of spontaneously beating guinea-pig atria with EC50 of 0.030 ug/mL.

物理化学性质&存储条件

分子量	456.5744
分子式	C26H36N2O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2H-3-Benzazepin-2-one, 3-[3-[[2-(3,4-dimethoxyphenyl)ethyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-

参考文献

1. Van Bogaert PP, et al. Eur J Pharmacol. 2003 Oct 8;478(2-3):161-71.

2. McGovern AE, et al. Br J Pharmacol. 2014 Aug;171(15):3633-50.

3. Gill CH, et al. Br J Pharmacol. 2004 Oct;143(3):411-21.

Zatebradine (UL-FS49)

生物&药学活性

物理化学性质&存储条件

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Zatebradine (UL-FS49)

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