ZINC-3573 racemate |CAS:1378183-16-4 Probechem Biochemicals

首页-小分子抑制剂&激动剂-GPCR-Mas-related G protein-coupled receptor (MRGPR)-ZINC-3573 racemate

Chemical Structure : ZINC-3573 racemate

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ZINC-3573 racemate (ZINC3573 racemate)

货号: PC-62228Not For Human Use, Lab Use Only.

ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases.
ZINC-3573 activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.

物理化学性质&存储条件

分子量	307.401
分子式	C18H21N5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Dimethyl-[1-(5-phenyl-pyrazolo[1,5-a]pyrimidin-7-yl)-pyrrolidin-3-yl]-amine

参考文献

1. Lansu K, et al. Nat Chem Biol. 2017 May;13(5):529-536.

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ZINC-3573 racemate (ZINC3573 racemate)

生物&药学活性

物理化学性质&存储条件

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ZINC-3573 racemate (ZINC3573 racemate)

生物&药学活性

物理化学性质&存储条件

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